17. Copper-catalyzed Conversion of Propargylic Bromodifluoroacetates to Trifluoromethanes

 
 

Ambler, B. R.; Peddi, S.; Altman, R. A.*

Synthesis 2014, 46, 1938–1946.

The development of efficient methods for accessing fluo­rinated functional groups is desirable. Herein, we report a two-step method that utilizes catalytic copper for the decarboxylative trifluoromethylation of propargyl bromodifluoroacetates is described. This protocol affords a mixture of propargyl trifluoromethanes and trifluoromethyl allenes.

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18. Metal-free Trifluoromethylation of Aromatic and Heteroaromatic Aldehydes and Ketones

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16. Decarboxylative Fluorination Strategies for Accessing Medicinally-Relevant Products